Synthesis and in vitro binding studies of piperazine-alkyl-naphthamides: Impact of homology and sulphonamide/carboxamide bioisosteric replacement on the affinity for 5-HT1A, alpha(2A), D4.2, D3 and D2L receptors
Résimont, Mélissa; Liégeois, Jean-François
2010 • In Bioorganic and Medicinal Chemistry Letters, 20, p. 5199-5202
Liégeois, Jean-François ; Université de Liège - ULiège > Département de pharmacie > Chimie pharmaceutique
Language :
English
Title :
Synthesis and in vitro binding studies of piperazine-alkyl-naphthamides: Impact of homology and sulphonamide/carboxamide bioisosteric replacement on the affinity for 5-HT1A, alpha(2A), D4.2, D3 and D2L receptors
B.L. Roth, D.L. Sheffler, and W.K. Kroeze Nat. Rev. Drug Disc. 3 2004 353
M.J. Marino, L.J.S. Knutsen, and M. Williams J. Med. Chem. 51 2008 1077
J. Ichikawa, I. Ishii, S. Bonaccorso, W.L. Fowler, I.A. O'Laughlin, and H.Y. Meltzer J. Neurochem. 76 2001 1521
P. Hertel, M.V. Fagerquist, and T.H. Svensson Science 286 1999 105
B.R. Chemel, B.L. Roth, B. Armbruster, V.J. Watts, and D.E. Nichols Psychopharmacology (Berlin) 188 2006 244
A. Graulich, M. Léonard, M. Résimont, X.-P. Huang, B.L. Roth, and J.-F. Liégeois Aust. J. Chem. 63 2010 56
J. Yoon, E. Yoo, J.-Y. Kim, A.N. Pae, H. Rhim, W.-K. Park, J.Y. Kong, and H.-Y. Park Choo Bioorg. Med. Chem. 16 2008 5405
P. Carato, A. Graulich, N. Jensen, B.L. Roth, and J.-F. Liégeois Bioorg. Med. Chem. Lett. 17 2007 1565
P. Carato, A. Graulich, N. Jensen, B.L. Roth, and J.-F. Liégeois Bioorg. Med. Chem. Lett. 17 2007 1570
F. Rodriguez, I. Rozas, J.E. Ortega, A.M. Erdozain, J.J. Meana, and L.F. Calldo J. Med. Chem. 52 2009 601
M. Pilla, S. Perachon, F. Sautel, F. Garrido, A. Mann, C.G. Wermuth, J.-C. Schwartz, B.J. Everitt, and P. Sokoloff Nature 400 1999 371
K. Wicke, and J. Garcia-Ladona Eur. J. Pharmacol. 424 2001 85
G. Campiani, S. Butini, F. Trotta, C. Fattorusso, B. Catalanotti, F. Aiello, S. Gemma, V. Nacci, E. Novellino, J. Ann Stark, A. Cagnotto, E. Fumagalli, F. Carnovali, L. Cervo, and T. Mennini J. Med. Chem. 46 2003 3822
A. Hackling, R. Ghosh, S. Perachon, A. Mann, H.-D. Höltje, C.G. Wermuth, J.-C. Schwartz, W. Sippl, P. Sokoloff, and H. Stark J. Med. Chem. 46 2003 3883
C.G. Wermuth The Practice of Medicinal Chemistry C.G. Wermuth, 2000 Academic Press 203
J.-F. Liégeois, G. Dive, L. Dupont, and J. Delarge Helv. Chim. Acta 74 1991 1764
J.-P. Fournier, R.C. Moreau, G. Narcisse, and P. Choay Eur. J. Med. Chem. 17 1982 81
A.J. Bojarski, B. Duszyńska, M. Kolaczkowski, P. Kowalski, and T. Kowalska Bioorg. Med. Chem. Lett. 23 2004 5863
R.A. Medina, J. Sallander, B. Benhamu, E. Porras, M. Campillo, L. Pardo, and M.L. Lopez-Rodriguez J. Med. Chem. 52 2009 2384
E. Yoo, J. Yoon, A.N. Pae, H. Rhim, W.-K. Park, J.Y. Kong, and H.-Y. Park Choo Bioorg. Med. Chem. 18 2010 1665
