Powers, J. C.; Zimmerman, M. In Design of Enzyme Inhibitors as Drugs; Sandler, M., Smith, H. J., Eds.; Oxford University Press: Oxford, 1989; pp 596-619.
Powers, J. C.; Harper, J. W. In Proteinase Inhibitors; Barett, A. J., Salvensen, G., Eds.; Elsevier: Amsterdam, 1986; pp 55-152.
Hlasta D.J., Pagani E.D. Ann. Rep. Med. Chem. 29:1994;195.
Janoff A. Am. Rev. Respir. Dis. 132:1985;417.
Demling R.H. Annu. Rev. Med. 46:1995;193.
Janoff A. Annu. Rev. Med. 36:1985;207.
Snider G.L. Drug. Dev. Res. 10:1987;235.
Nadel J.A. Am. Rev. Respir. Dis. 14:1991;S48.
Rai R., Katzenellenbogen J.A. J. Med. Chem. 35:1992;4297.
Rai R., Katzenellenbogen J.A. J. Med. Chem. 35:1992;4150.
Katzenellenbogen J.A., Rai R., Dai W. Bioorg. Med. Chem. Lett. 2:1992;1399.
Finke P.E., Ashe B.M., Knight W.B., Maycock A.L., Navia M.A., Shah S.K., Thompson K.R., Underwood D.J., Weston H., Zimmerman M., Doherty J.B. J. Med. Chem. 33:1990;2522.
Finke P.E., Shah S.K., Fletcher D.S., Ashe B.M., Brause K.A., Chandler G.O., Dellea P.S., Hand K.M., Maycock A.L., Osinga D.G., Underwood D.J., Weston H., Davies P. J. Med. Chem. 38:1995;2449.
Knight W.B., Green B.G., Chabin R.M., Gale P., Maycock A.L., Weston H., Kuo D.W., Westler W.M., Dorn C.P., Finke P.E., Hagmann W.K., Hale J.J., Liesh J., MacCoss M., Navia M.A., Shah S.K., Underwood D., Doherty J.B. Biochemistry. 31:1992;8160.
Wakselman M., Joyeau R., Kobaiter R., Bogetto N., Vergely I., Maillard J., Okochi V., Montagne J.J., Reboud-Ravaux M. FEBS Lett. 282:1991;377.
Groutas W.C., Houser-Archield N., Chong L.S., Venkataraman R., Epp J.B., Huang H., McClenahan J.J. J. Med. Chem. 36:1993;3178.
Desai R.C., Court J.C., Ferguson E., Gordon R.J., Hlasta D.J., Dunlap R.P., Franke C.A. J. Med. Chem. 38:1995;1571.
Krantz A., Spencer R.W., Tam T.F., Liak T.J., Copp L.J., Thomas E.M., Rafferty S.P. J. Med. Chem. 33:1990;464.
Uejima Y., Kokubo M., Oshida J., Kawabata H., Kato Y., Fujii K. Pharmacol. Exp. Ther. 265:1993;516.
Hernandez M.A., Powers J.C., Glinski J., Oleksyszyn J., Vijayalakshmi J., Meyer E.F. Jr. J. Med. Chem. 35:1992;1121.
Kam C.M., Kerrigan J.E., Plaskon R.R., Duffy E.J., Lollar P., Suddath F.L., Powers J.C. J. Med. Chem. 37:1994;1298.
Kerrigan J.E., Oleksyszyn J., Kam C.M., Selzler J., Powers J.C. J. Med. Chem. 38:1995;544.
Béchet J.-J., Dupaix A., Yon J., Wakselman M., Robert J.-L., Vilkas M. Eur. J. Biochem. 35:1973;527.
Mor A., Maillard J., Favreau C., Reboud-Ravaux M. Biochim. Biophys. Acta. 1038:1990;119.
Groutas W.C., Kuang R., Venkataraman R. Biochem. Biophys. Res. Commun. 198:1994;341.
Groutas W.C., Kuang R., Venkataraman R., Epp J.B., Ruan S., Prakash O. Biochemistry. 36:1997;4739.
Pochet L., Doucet C., Schynts M., Thierry N., Boggetto N., Pirotte B., Jiang K.-Y., Masereel B., de Tullio P., Delarge J., Reboud-Ravaux M. J. Med. Chem. 39:1996;2579.
Wakselman M. Nouv. J. Chim. 7:1983;439.
Dive G., Dehareng D., Peeters D. Int. J. Quant. Chem. 58:1996;85.
Boggetto N., Vilain A.C., Montagne J.J., Reboud-Ravaux M., Mazaleyrat J.P., Xie J., Wakselman M. Bull. Soc. Chim. Fr. 131:1994;152.
Joyeau R., Felk A., Guilaume S., Wakselman M., Vergely I., Doucet C., Boggetto N., Reboud-Ravaux M. J. Pharm. Pharmacol. 48:1996;1218.
Doucet C., Vergely I., Reboud-Ravaux M., Guilhem J., Kobaiter R., Joyeau R., Wakselman M. Tetrahedron: Asymmetry. 8:1997;739.
Doucet C., Pochet L., Thierry N., Pirotte B., Delarge J., Reboud-Ravaux M. J. Med. Chem. 42:1999;4161.
kinact/KI for 52, 53 and 54 was 48,100, 762,700, 330 M-1 s-1, respectively. See ref 28.
Bowden, J.; Hanson, M. J.; Taylor, G. R. J. Chem. Soc. 1968, 174.
Lippold B.C., Garett E.R. J. Pharm. Sci. 60:1971;1019.
Wakselman M., Xie J., Mazaleyrat J.-P., Bogetto N., Vilain A.-C., Montagne J.-J., Reboud-Ravaux M. J. Med. Chem. 36:1993;1539.
Silverman, R. B. In Mechanism-Based Enzyme Inactivation: Chemistry and Enzymology; CRC Press: Boca Raton, FL, 1988; Vol. 1, pp 22-23.
Tatewaki H., Huzinaga S. J. Comp. Chem. 1:1980;205.
Dive G., Dehareng D., Ghuysen J.M. Theoret. Chim. Acta. 85:1993;409.
Frisch, M. J.; Trucks, G. W.; Schlegel, H. B.;Gill, P. M. W.; Johnson, B. G.; Robb, M. A.; Cheeseman, J. R.; Keith, T.; Petersson, G. A.; Montgomery, J. A.; Raghavachari, K.; Al-Laham, M. A.; Zakrzewski, V. G.; Ortiz, J. V.; Foresman, J. B.; Cioslowski, J.; Stefanov, B. B.; Nanayakkara, A.; Challacombe, M.; Peng, C. Y.; Ayala, P. Y.; Chen, W.; Wong, M. W.; Andres, J. L.; Replogle, E. S.; Gomperts, R.; Martin, R. L.; Fox, D. J.; Binkley, J. S.; Defrees, D. J.; Baker, J.; Stewart, J. P.; Head-Gordon, M.; Gonzalez, C.; Pople, J. A. Gaussian 94, Revision D.4; Pittsburgh, PA, 1995.
