Aguilar-Bryan L., Bryan J. (1999) Molecular biology of adenosine triphosphate-sensitive potassium channels. Endocrine Rev. 20:101-135.
Antoine M.-H., Berkenboom G., Fang Z.Y., Fontaine J., Herchuelz A., Lebrun P. (1992) Mechanical and ionic response of rat aorta to diazoxide. Eur. J. Pharmacol. 216:299-306.
Antoine M.-H., Hermann M., Herchuelz A., Lebrun P. (1991) Ionic and secretory response of pancreatic islet cells to minoxidil sulfate. J. Pharmacol. Exp. Ther. 258:286-291.
Antoine M.-H., Hermann M., Herchuelz A., Lebrun P. (1993) Sodium nitroprusside inhibits glucose-induced insulin release by activating ATP-sensitive K+ channels. Biochim. Biophys. Acta. 1175:293-301.
Ashcroft S.J.H., Ashcroft F.M. (1990) Properties and functions of ATP-sensitive K-channels. Cell. Signal. 2:197-214.
Ashcroft F.M., Gribble F.M. (1998) Correlating structure and function in ATP-sensitive K+ channels. TINS 21:288-294.
Ashcroft F.M., Harrison D.E., Ashcroft S.J.H. (1984) Glucose induces closure of single potassium channels in isolated rat pancreatic β-cells. Nature 312:446-448.
Ashcroft F.M., Rorsman P. (1989) Electrophysiology of the pancreatic B-cell. Prog. Biophys. Mol. Biol. 54:87-143.
Ashford M.L.J., Sturgess N.C., Trout N.J., Gardner N.J., Hales C.N. (1988) Adenosine-5′-triphosphate-sensitive ion channels in neonatal rat cultured central neurones. Pflügers Arch. 412:297-304.
Bandoli G., Nicolini M. (1977) Crystal and molecular structure of diazoxide, an antihypertensive agent. J. Cryst. Mol. Struct. 7:229-240.
Cloux J.L., Crommen J., Delarge J., Pirard M.L., Thunus L. (1988) Tentative de détermination de la constante fragmentaire (f) du groupement sulfonylurée. J. Pharm. Belg. 43:141-151.
Cook D.L., Hales C.N. (1984) Intracellular ATP directly blocks K+ channels in pancreatic β-cells. Nature 311:271-273.
De Tullio P., Pirotte B., Lebrun P., Fontaine J., Dupont L., Antoine M.-H., Ouedraogo R., Khelili S., Maggetto C., Masereel B., Diouf O., Podona T., Delarge J. (1996) 3- and 4-substituted 4H-Pyrido[4,3-e]-1,2,4-thiadiazine 1,1-dioxides as potassium channel openers: Synthesis, pharmacological evaluation, and structure-activity relationships. J. Med. Chem. 39:937-948.
Desai K., Desai C.M. (1967) Direct synthesis of 4-hydroxyquinolines using polyphosphoric acid. Indian J. Chem. 5:170-171.
Edwards G., Weston A.H. (1993) The pharmacology of ATP-sensitive potassium channels. Ann. Rev. Pharmacol. Toxicol. 33:597-637.
Franchi G., Vigni P. (1967) Nuovi composti chinolinici fluorurati ad azione antibatterica. Il Farmaco 22:923-929.
Gerber J.G., Nies A.S. (1990) Antihypertensive agents and the drug therapy of hypertension. The pharmacological basis of therapeutics (8th ed.) , eds. A.G. Goodman-Gilman, T.W. Rall, A.S. Nies & P. Taylor. New York: Pergamon Press; 784-805.
Hamill O.P., Marty A., Neher E., Sakmann B., Sigworth F.J. (1981) Improved patch-clamp techniques for high-resolution current recording from cells and cell-free membrane patches. Pflügers Archiv. 391:85-100.
Hansch C., Leo A., Unger S.H., Kim K.H., Nikaitani D., Lien E.J. (1973) Aromatic substituent constants for structure-activity correlations. J. Med. Chem. 16:1207-1216.
Henquin J.C., Debuyser A., Drews G., Plant T.D. (1992) Regulation of K+ permeability and membrane potential in insulin secreting cells. Nutrient Regulation of Insulin Secretion , ed. Flatt P.R. Portland Press Ltd, London; 173-191.
Inoue I., Nagase H., Kishi K., Higuti T. (1991) ATP-sensitive K+ channel in the mitochondrial inner membrane. Nature 352:244-247.
Jakobsen P., Treppendahl S. (1979) The structure of 1,2,4-benzothiadiazine-1, 1-dioxides. Tetrahedron 35:2151-2153.
Kane C., Shepherd R.M., Squires P.E., Johnson P.R.V., James R.F.L., Milla P.J., Aynsley-Green A., Lindley K.J., Dunne M.J. (1996) Loss of functional KATP channels in β-cells causes persistent hyperinsulinaemic hypoglycaemia of infancy. Nature Med. 2:1344-1347.
Katritzky A.R. (1985) Structure of 6-membered rings. Handbook of heterocyclic chemistry , ed. Katritzky A.R. Oxford: Pergamon Press; 23-51.
Lacy P.E., Kostianowsky M. (1967) Method for the isolation of intact islets of Langerhans from the rat pancreas. Diabetes 16:35-39.
Lebrun P., Antoine M.-H., Herchuelz A. (1992) Minireview: K+ channel openers and insulin release. Life Sci. 51:795-806.
Lebrun P., Antoine M.-H., Ouedraogo R., Kane C., Dunne M., Hermann M., Herchvelz A., Masereel B., Delarge J., De Tullio P., Pirotte B. (1996) Activation of ATP-dependent K+ channels and inhibition of insulin release: Effect of BPDZ 62. J. Pharmacol. Exp. Ther. 277:156-162.
Lebrun P., Arkhammar P., Antoine M.-H., Nguyen Q.-A., Bondo Hansen J., Pirotte B. (2000) A potent diazoxide analogue activating ATP-sensitive K+ channels and inhibiting insulin release. Diabetologia 43:723-732.
Lebrun P., Atwater I. (1985) Effects of the calcium channel agonist, BAY K 8644, on electrical activity in mouse pancreatic B-cells. Biophys. J. 48:919-930.
Lebrun P., Devreux V., Hermann M., Herchuelz A. (1989) Similarities between the effects of pinacidil and diazoxide on ionic and secretory events in rat pancreatic islets. J. Pharmacol. Exp. Ther. 250:1011-1018.
Lebrun P., Fang Z.Y., Antoine M.-H., Herchuelz A., Hermann M., Berkenboom G., Fontaine J. (1990) Hypoglycemic sulfonylureas antagonize the effects of cromakalim and pinacidil on 86Rb fluxes and contractile activity in the rat aorta. Pharmacology 41:36-48.
Lebrun P., Malaisse W.J., Herchuelz A. (1982) Evidence for two distinct modalities of Ca2+ influx into pancreatic B cell. Am. J. Physiol. 242.
Leclercq-Meyer V., Marchand J., Woussen-Colle M.C., Giroix M.H., Malaisse W.J. (1985) Multiple effects of leucine on glucagon, insulin and somatostatin secretion from the perifused rat pancreas. Endocrinology 116:1168-1174.
Macfarlane W.M., O'Brien R.E., Barnes P.D., Shepherd R.M., Cosgrove K.E., Lindley K.J., Aynsley-Green A., James R.F.L., Docherty K., Dunne M.J. (2000) Sulphonylurea receptor 1 and Kit 6.2 expression in the novel human insulin-secreting cell line NES2Y. Diabetes 49:953-960.
Magnon M., Calderone V., Floch A., Cavero I. (1998) Influence of depolarization on vasorelaxant potency and efficacy of Ca2+ entry blockers, K+ channel openers, nitrate derivatives, salbutamol and papaverine in rat aortic rings. Naunyn-Schmiedeberg's Arch. Pharmacol. 358:452-463.
Malaisse W.J., Boschero A.C., Kawazu S., Hutton J.C. (1978) The stimulus secretion coupling of glucose-induced insulin release. XXVII. Effect of glucose on K+ fluxes in isolated islets. Pflügers Arch. 373:237-242.
Malaisse W.J., Lebrun P. (1990) Mechanisms of sulfonylurea-induced insulin release. Diabetes Care 13:9-17.
Mallams A.K., Israelstam S.S. (1964) The reaction between β-keto esters and arylamines in the presence of polyphosphoric acid. II. Ethyl acetoacetate and its α-alkyl derivatives and arylamines. J. Org. Chem. 29:3548-3554.
Miki T., Nagashima K., Seino S. (1999) The structure and function of the ATP-sensitive K+ channel in insulin-secreting pancreatic β-cells. J. Mol. Endocrinol. 22:113-123.
Nichols C.G., Lederer W.J. (1991) Adenosine triphosphate-sensitive potassium channels in the cardiovascular system. Am. J. Physiol. 261.
Noma A. (1983) ATP-regulated K+ channels in cardiac muscle. Nature 305:147-148.
Pipeleers D.G., In'T Veld P.A., Van De Winkel M., Maes E., Schuit F.C., Gepts W. (1985) A new in vitro model for the study of pancreatic α and β cells. Endocrinology 117:806-816.
Pirotte B., Ouedraogo R., De Tullio P., Khelili S., Somers F., Boverie S., Dupont L., Fontaine J., Damas J., Lebrun P. (2000) 3-Alkylamino-4H-pyrido[2,3-e]-1,2,4-thiadiazine 1,1-dioxides structurally related to diazoxide and pinacidil as potassium channel openers acting on vascular smooth muscle cells: Design, synthesis, and pharmacological evaluation. J. Med. Chem. 43:1456-1466.
Quast U. (1993) Do the K+ channel openers relax smooth muscle by opening K+ channels?. TiPS 14:332-337.
Quast U., Baumlin Y. (1988) Comparison of the effluxes of 42K+ and 86Rb+ elicited by cromakalim (BRL 34915) in tonic and phasic vascular tissue. Naunyn-Schmiedeberg's Arch. Pharmacol. 338:319-326.
Quast U., Cook N.S. (1989) In vitro and in vivo comparison of two K+ channel openers, diazoxide and cromakalim, and their inhibition by glibenclamide. J. Pharmacol. Exp. Ther. 250:261-271.
Rorsman P., Trube G. (1985) Glucose dependent K+ channels in pancreatic β-cells are regulated by intracellular ATP. Pflügers Archiv. 405:305-309.
Seino S. (1999) ATP-sensitive potassium channels: A model of heteromultimeric potassium channel/receptor assemblies. Ann. Rev. Physiol. 61:337-362.
Suzuki M., Kotake K., Fujikura K., Inagaki N., Suzuki T. (1997) Kir 6.1: A possible subunit of ATP-sensitive K+ channels in mitochondria. Biochem. Biophys. Res. Commun. 241:693-697.
Szewczyk A., Marban E. (1999) Mitochondria: A new target for K+ channel openers?. Trends Pharmacol. Sci. 20:157-161.
Tucker S.J., Gribble F.M., Zhao C., Trapp S., Ashcroft F.M. (1997) Truncation of Kir 6.2 produces ATP-sensitive K+-channels in the absence of the sulphonylurea receptor. Nature 378:179-183.
Verkarre V., Fournet J.C., De Lonlay P., Gross-Morand M.S., Devillers M., Rahier J., Brunelle F., Robert J.J., Nihoul-Fekete C., Saudubray J.M., Junien C. (1998) Paternal mutation of the sulfonylurea receptor (SUR1) gene and maternal loss of 11p15 imprinted genes lead to persistent hyperinsulinism in focal adenomatous hyperplasia. J. Clin. Invest. 102:1286-1291.
