Synthesis of [18F]4-(4-fluorophenyl)-1,2,4-triazole-3,5-dione: an agent for specific radiolabelling of tyrosine

Flagothier, Jessica; Warnier, Corentin; Dammicco, Sylvestre; Lemaire, Christian; Luxen, André

doi:10.1039/c3ra44666b

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Synthesis of [18F]4-(4-fluorophenyl)-1,2,4-triazole-3,5-dione: an agent for specific radiolabelling of tyrosine

Flagothier, Jessica; Warnier, Corentin; Dammicco, Sylvestre et al.

2013 • In RSC Advances, 3, p. 24936

Peer Reviewed verified by ORBi

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https://hdl.handle.net/2268/164270

DOI
10.1039/c3ra44666b

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Keywords :

fluorine-18; radiosynthesis; tyrosine

Abstract :

[en] We developed a new [18F] prosthetic group, the [18F]4-(4-fluorophenyl)-1,2,4-triazole-3,5-dione ([18F]FPTAD), used for its specific ligation with tyrosine-containing peptides or protein in order to develop a new and versatile radiolabelling technique that could provide a useful tool for new developments in PET imaging.

Research Center/Unit :

GIGA CRC (Cyclotron Research Center) In vivo Imaging-Aging & Memory - ULiège

Disciplines :

Chemistry

Author, co-author :

Flagothier, Jessica ; Université de Liège - ULiège > Département de chimie (sciences) > Chimie organique de synthèse

Warnier, Corentin ; Université de Liège - ULiège > Centre de recherches du cyclotron

Dammicco, Sylvestre ; Université de Liège - ULiège > Département de chimie (sciences) > Chimie organique de synthèse

Lemaire, Christian ; Université de Liège - ULiège > Centre de recherches du cyclotron

Luxen, André ; Université de Liège - ULiège > Département de chimie (sciences) > Chimie organique de synthèse

Language :

English

Title :

Synthesis of [18F]4-(4-fluorophenyl)-1,2,4-triazole-3,5-dione: an agent for specific radiolabelling of tyrosine

Alternative titles :

[fr] Synthèse du [18F]4-(4-fluorophenyl)-1,2,4-triazole-3,5-dione: un agent pour le marquage spécifique des tyrosines

Publication date :

10 October 2013

Journal title :

RSC Advances

eISSN :

2046-2069

Publisher :

Royal Society of Chemistry Publishing, Cambridge, United Kingdom

Volume :

Pages :

24936

Peer reviewed :

Peer Reviewed verified by ORBi

Available on ORBi :

since 16 March 2014

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